Skip to main content

Lund University Publications

LUND UNIVERSITY LIBRARIES

Arynes in the Monoarylation of Unprotected Carbohydrate Amines

Pal, Kumar Bhaskar ; Mahanti, Mukul LU and Nilsson, Ulf J. LU (2018) In Organic Letters 20(3). p.616-619
Abstract

A CsF-mediated method has been developed for the N-arylation of amino sugars that affords good to excellent yields of arylated products under mild conditions involving the in situ generation of arynes. The reaction conditions tolerate a variety of common carbohydrate protecting groups and also performs exceptionally well on unprotected amino sugar derivatives. The reactions are scalable in moderate to good yields with broad scope.

Please use this url to cite or link to this publication:
author
; and
organization
publishing date
type
Contribution to journal
publication status
published
subject
in
Organic Letters
volume
20
issue
3
pages
4 pages
publisher
The American Chemical Society (ACS)
external identifiers
  • pmid:29359567
  • scopus:85041603885
ISSN
1523-7060
DOI
10.1021/acs.orglett.7b03741
language
English
LU publication?
yes
id
66fb37bb-e697-48a1-9afc-d5ceebfc11c1
date added to LUP
2018-02-21 10:03:56
date last changed
2024-03-18 05:24:27
@article{66fb37bb-e697-48a1-9afc-d5ceebfc11c1,
  abstract     = {{<p>A CsF-mediated method has been developed for the N-arylation of amino sugars that affords good to excellent yields of arylated products under mild conditions involving the in situ generation of arynes. The reaction conditions tolerate a variety of common carbohydrate protecting groups and also performs exceptionally well on unprotected amino sugar derivatives. The reactions are scalable in moderate to good yields with broad scope.</p>}},
  author       = {{Pal, Kumar Bhaskar and Mahanti, Mukul and Nilsson, Ulf J.}},
  issn         = {{1523-7060}},
  language     = {{eng}},
  month        = {{02}},
  number       = {{3}},
  pages        = {{616--619}},
  publisher    = {{The American Chemical Society (ACS)}},
  series       = {{Organic Letters}},
  title        = {{Arynes in the Monoarylation of Unprotected Carbohydrate Amines}},
  url          = {{http://dx.doi.org/10.1021/acs.orglett.7b03741}},
  doi          = {{10.1021/acs.orglett.7b03741}},
  volume       = {{20}},
  year         = {{2018}},
}