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2017
Mark Structural Basis for Potency and Promiscuity in Poly(ADP-ribose) Polymerase (PARP) and Tankyrase Inhibitors
Thorsell, Ann-Gerd ; Ekblad, Torun ; Karlberg, Tobias ^LU ; Löw, Mirjam ; Pinto, Ana Filipa ; Trésaugues, Lionel ; Moche, Martin ; Cohen, Michael S and Schüler, Herwig ^LU (2017) In Journal of Medicinal Chemistry 60(4). p.1262-1271
- Contribution to journal › Article
2015
Mark Tankyrase 1 Inhibitors with Drug-like Properties Identified by Screening a DNA-Encoded Chemical Library
Samain, Florent ; Ekblad, Torun ; Mikutis, Gediminas ; Zhong, Nan ; Zimmermann, Mauro ; Nauer, Angela ; Bajic, Davor ; Decurtins, Willy ; Scheuermann, Jörg and Brown, Peter J , et al. (2015) In Journal of Medicinal Chemistry 58(12). p.9-5143
- Contribution to journal › Article
Mark Identification of structure-activity relationships from screening a structurally compact DNA-encoded chemical library
Franzini, Raphael M ; Ekblad, Torun ; Zhong, Nan ; Wichert, Moreno ; Decurtins, Willy ; Nauer, Angela ; Zimmermann, Mauro ; Samain, Florent ; Scheuermann, Jörg and Brown, Peter J , et al. (2015) In Angewandte Chemie (International edition) 54(13). p.31-3927
- Contribution to journal › Article
2014
Mark Design, synthesis, crystallographic studies, and preliminary biological appraisal of new substituted triazolo[4,3-b]pyridazin-8-amine derivatives as tankyrase inhibitors
Liscio, Paride ; Carotti, Andrea ; Asciutti, Stefania ; Karlberg, Tobias ^LU ; Bellocchi, Daniele ; Llacuna, Laura ; Macchiarulo, Antonio ; Aaronson, Stuart A ; Schüler, Herwig ^LU and Pellicciari, Roberto , et al. (2014) In Journal of Medicinal Chemistry 57(6). p.12-2807
- Contribution to journal › Article
2012
Mark Family-wide chemical profiling and structural analysis of PARP and tankyrase inhibitors
Wahlberg, Elisabet ; Karlberg, Tobias ^LU ; Kouznetsova, Ekaterina ; Markova, Natalia ^LU ; Macchiarulo, Antonio ; Thorsell, Ann-Gerd ; Pol, Ewa ; Frostell, Åsa ; Ekblad, Torun and Öncü, Delal , et al. (2012) In Nature Biotechnology 30(3). p.8-283
- Contribution to journal › Article
2010
Mark Structural basis for the interaction between tankyrase-2 and a potent Wnt-signaling inhibitor
Karlberg, Tobias ^LU ; Markova, Natalia ^LU ; Johansson, Ida ^LU ; Hammarström, Martin ; Schütz, Patrick ; Weigelt, Johan and Schüler, Herwig ^LU (2010) In Journal of Medicinal Chemistry 53(14). p.5-5352
- Contribution to journal › Article