Peptidyl diazomethylketones as cysteine protease inhibitors structurally based upon the inhibitory centers of cystatins
(2001) In Polish Journal of Chemistry 75(6). p.831-837- Abstract
- Six new putative cysteine protease inhibitors based upon sequences of the N-terminal binding fragments of rat cystatin A, bovine cystatin C and human cystatins D and S were synthesized, inhibitory activities of these compounds against papain and bovine cathepsin B were tested. Additionally, agar well diffusion test of their antibacterial activity against Streptococcus pyogenes was performed.
Please use this url to cite or link to this publication:
https://lup.lub.lu.se/record/1119163
- author
- Kasprzykowski, F.
; Kasprzykowska, R.
; Kania, P.
; Plucinska, K.
; Grubb, Anders
LU
; Abrahamson, Magnus LU and Schalen, C.
- organization
- publishing date
- 2001
- type
- Contribution to journal
- publication status
- published
- subject
- in
- Polish Journal of Chemistry
- volume
- 75
- issue
- 6
- pages
- 831 - 837
- publisher
- Polish Chemical Society
- external identifiers
-
- wos:000169182500007
- scopus:0035534834
- ISSN
- 0137-5083
- language
- English
- LU publication?
- yes
- id
- c79701bc-b10d-4cf8-8db8-0ca1c60be490 (old id 1119163)
- date added to LUP
- 2016-04-01 16:10:47
- date last changed
- 2023-01-04 21:53:40
@article{c79701bc-b10d-4cf8-8db8-0ca1c60be490, abstract = {{Six new putative cysteine protease inhibitors based upon sequences of the N-terminal binding fragments of rat cystatin A, bovine cystatin C and human cystatins D and S were synthesized, inhibitory activities of these compounds against papain and bovine cathepsin B were tested. Additionally, agar well diffusion test of their antibacterial activity against Streptococcus pyogenes was performed.}}, author = {{Kasprzykowski, F. and Kasprzykowska, R. and Kania, P. and Plucinska, K. and Grubb, Anders and Abrahamson, Magnus and Schalen, C.}}, issn = {{0137-5083}}, language = {{eng}}, number = {{6}}, pages = {{831--837}}, publisher = {{Polish Chemical Society}}, series = {{Polish Journal of Chemistry}}, title = {{Peptidyl diazomethylketones as cysteine protease inhibitors structurally based upon the inhibitory centers of cystatins}}, volume = {{75}}, year = {{2001}}, }