A meroterpenoid NF-kappa B inhibitor and drimane sesquiterpenoids from asafetida
(2006) In Journal of Natural Products 69(7). p.1101-1104- Abstract
- Investigation of an acetone extract from asafetida afforded two drimane sesquiterpene dienones (fetidones A and B, 1a,b) and several known sesquiterpene coumarin ethers, one of which (8-acetoxy-5-hydroxyumbelliprenin, 2a) showed potent and specific NF-kappa B-inhibiting properties. This, coupled to a negligible cytotoxicity, qualifies 2a as a new anti-inflammatory chemotype, and its occurrence in asafetida might rationalize the use of this gum resin to alleviate and prevent colon inflammatory disturbances.
Please use this url to cite or link to this publication:
https://lup.lub.lu.se/record/399493
- author
- Appendino, Giovanni ; Maxia, Lucia ; Bascope, Marcelo LU ; Houghton, Peter J. ; Sanchez-Duffhues, Gonzalo ; Munoz, Eduardo and Sterner, Olov LU
- organization
- publishing date
- 2006
- type
- Contribution to journal
- publication status
- published
- subject
- in
- Journal of Natural Products
- volume
- 69
- issue
- 7
- pages
- 1101 - 1104
- publisher
- The American Chemical Society (ACS)
- external identifiers
-
- pmid:16872156
- wos:000239336000028
- scopus:33747421726
- pmid:16872156
- ISSN
- 0163-3864
- DOI
- 10.1021/np0600954
- language
- English
- LU publication?
- yes
- additional info
- The information about affiliations in this record was updated in December 2015. The record was previously connected to the following departments: Organic chemistry (S/LTH) (011001240)
- id
- 0b2c1138-0d7a-42e4-975e-dc60c199adab (old id 399493)
- date added to LUP
- 2016-04-01 16:07:07
- date last changed
- 2022-02-20 03:23:16
@article{0b2c1138-0d7a-42e4-975e-dc60c199adab, abstract = {{Investigation of an acetone extract from asafetida afforded two drimane sesquiterpene dienones (fetidones A and B, 1a,b) and several known sesquiterpene coumarin ethers, one of which (8-acetoxy-5-hydroxyumbelliprenin, 2a) showed potent and specific NF-kappa B-inhibiting properties. This, coupled to a negligible cytotoxicity, qualifies 2a as a new anti-inflammatory chemotype, and its occurrence in asafetida might rationalize the use of this gum resin to alleviate and prevent colon inflammatory disturbances.}}, author = {{Appendino, Giovanni and Maxia, Lucia and Bascope, Marcelo and Houghton, Peter J. and Sanchez-Duffhues, Gonzalo and Munoz, Eduardo and Sterner, Olov}}, issn = {{0163-3864}}, language = {{eng}}, number = {{7}}, pages = {{1101--1104}}, publisher = {{The American Chemical Society (ACS)}}, series = {{Journal of Natural Products}}, title = {{A meroterpenoid NF-kappa B inhibitor and drimane sesquiterpenoids from asafetida}}, url = {{http://dx.doi.org/10.1021/np0600954}}, doi = {{10.1021/np0600954}}, volume = {{69}}, year = {{2006}}, }