Structural insights into urocanate reductase using room-temperature X-ray crystallography
(2026) In Acta Crystallographica Section D: Structural Biology 82. p.603-614- Abstract
Urocanate reductase (UrdA) is a bacterial enzyme that converts urocanic acid to imidazole propionate. Its catalytic residue Arg411 undergoes a large conformational change in the substrate-bound versus product-bound states. In contrast to previously studied cryo-conditions, the room-temperature X-ray data of UrdA presented here show that the occupancy distribution of Arg411 is affected by crystal cryocooling. We further provide evidence that a phosphate ion stabilizes the substrate complex and can bias the conformation of Arg411. Both room-temperature and cryogenic X-ray datasets were essential to elucidate the dynamic nature of the UrdA active site, highlighting the importance of collecting data at both temperatures, as each may reveal... (More)
Urocanate reductase (UrdA) is a bacterial enzyme that converts urocanic acid to imidazole propionate. Its catalytic residue Arg411 undergoes a large conformational change in the substrate-bound versus product-bound states. In contrast to previously studied cryo-conditions, the room-temperature X-ray data of UrdA presented here show that the occupancy distribution of Arg411 is affected by crystal cryocooling. We further provide evidence that a phosphate ion stabilizes the substrate complex and can bias the conformation of Arg411. Both room-temperature and cryogenic X-ray datasets were essential to elucidate the dynamic nature of the UrdA active site, highlighting the importance of collecting data at both temperatures, as each may reveal distinct conformational states.
(Less)
- author
- Aggarwal, Swati
LU
; Gurav, Nitisha
LU
; Oksanen, Esko
LU
; Lindkvist-Petersson, Karin
LU
and Venskutonytė, Raminta
LU
- organization
- publishing date
- 2026-06
- type
- Contribution to journal
- publication status
- published
- subject
- keywords
- active-site anion interactions, room-temperature crystallography, urocanate reductase
- in
- Acta Crystallographica Section D: Structural Biology
- volume
- 82
- pages
- 12 pages
- publisher
- John Wiley & Sons Inc.
- external identifiers
-
- pmid:42083916
- scopus:105040691551
- ISSN
- 2059-7983
- DOI
- 10.1107/S2059798326003360
- language
- English
- LU publication?
- yes
- id
- de8c843f-c1d4-4869-a0c9-50c9c05e0f1e
- date added to LUP
- 2026-07-03 10:00:25
- date last changed
- 2026-08-14 14:08:20
@article{de8c843f-c1d4-4869-a0c9-50c9c05e0f1e,
abstract = {{<p>Urocanate reductase (UrdA) is a bacterial enzyme that converts urocanic acid to imidazole propionate. Its catalytic residue Arg411 undergoes a large conformational change in the substrate-bound versus product-bound states. In contrast to previously studied cryo-conditions, the room-temperature X-ray data of UrdA presented here show that the occupancy distribution of Arg411 is affected by crystal cryocooling. We further provide evidence that a phosphate ion stabilizes the substrate complex and can bias the conformation of Arg411. Both room-temperature and cryogenic X-ray datasets were essential to elucidate the dynamic nature of the UrdA active site, highlighting the importance of collecting data at both temperatures, as each may reveal distinct conformational states.</p>}},
author = {{Aggarwal, Swati and Gurav, Nitisha and Oksanen, Esko and Lindkvist-Petersson, Karin and Venskutonytė, Raminta}},
issn = {{2059-7983}},
keywords = {{active-site anion interactions; room-temperature crystallography; urocanate reductase}},
language = {{eng}},
pages = {{603--614}},
publisher = {{John Wiley & Sons Inc.}},
series = {{Acta Crystallographica Section D: Structural Biology}},
title = {{Structural insights into urocanate reductase using room-temperature X-ray crystallography}},
url = {{http://dx.doi.org/10.1107/S2059798326003360}},
doi = {{10.1107/S2059798326003360}},
volume = {{82}},
year = {{2026}},
}