The p75 neurotrophin receptor enhances HIF-dependent signaling in glioma
(2018) In Experimental Cell Research 371(1). p.122-129- Abstract
Tumor hypoxia is associated with several features of aggressive glioma growth, including migration, invasion, and stemness. Most of the cellular adaptation to hypoxia is mediated by the hypoxia-inducible factors HIF-1α and HIF-2α, but regulation of these factors by both oxygen-dependent and –independent mechanisms in brain tumors is only partially understood. Here, we show that the p75 neurotrophin receptor (p75NTR) is stabilized at hypoxia in murine glioma in vivo, as well as in primary human glioma cultures in vitro. Expression of p75NTR resulted in increased stabilization of HIF-1α and HIF-2α, and RNAi or pharmacologic targeting of p75NTR diminished HIF stabilization and HIF-dependent signaling at... (More)
Tumor hypoxia is associated with several features of aggressive glioma growth, including migration, invasion, and stemness. Most of the cellular adaptation to hypoxia is mediated by the hypoxia-inducible factors HIF-1α and HIF-2α, but regulation of these factors by both oxygen-dependent and –independent mechanisms in brain tumors is only partially understood. Here, we show that the p75 neurotrophin receptor (p75NTR) is stabilized at hypoxia in murine glioma in vivo, as well as in primary human glioma cultures in vitro. Expression of p75NTR resulted in increased stabilization of HIF-1α and HIF-2α, and RNAi or pharmacologic targeting of p75NTR diminished HIF stabilization and HIF-dependent signaling at hypoxia. Consequentially, p75NTR inhibition resulted in decreased migration, invasion, and stemness in response to hypoxia, suggesting that p75NTR is a central regulator of hypoxia-induced glioma aggressiveness. Together, our findings support the literature that identifies p75NTR as a potential therapeutic target in brain tumors.
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- author
- Tong, Bei LU ; Pantazopoulou, Vasiliki LU ; Johansson, Elinn LU and Pietras, Alexander LU
- organization
- publishing date
- 2018-10-01
- type
- Contribution to journal
- publication status
- published
- subject
- keywords
- Glioblastoma multiforme, HIF-1α, HIF-2α, Hypoxia, P75 neurotrophin receptor, Stemness
- in
- Experimental Cell Research
- volume
- 371
- issue
- 1
- pages
- 8 pages
- publisher
- Academic Press
- external identifiers
-
- pmid:30092219
- scopus:85051059075
- ISSN
- 0014-4827
- DOI
- 10.1016/j.yexcr.2018.08.002
- language
- English
- LU publication?
- yes
- id
- 864cc259-d1cc-4da3-89ad-b1be0f4c3c98
- date added to LUP
- 2018-09-12 14:05:46
- date last changed
- 2024-10-15 07:00:50
@article{864cc259-d1cc-4da3-89ad-b1be0f4c3c98, abstract = {{<p>Tumor hypoxia is associated with several features of aggressive glioma growth, including migration, invasion, and stemness. Most of the cellular adaptation to hypoxia is mediated by the hypoxia-inducible factors HIF-1α and HIF-2α, but regulation of these factors by both oxygen-dependent and –independent mechanisms in brain tumors is only partially understood. Here, we show that the p75 neurotrophin receptor (p75<sup>NTR</sup>) is stabilized at hypoxia in murine glioma in vivo, as well as in primary human glioma cultures in vitro. Expression of p75<sup>NTR</sup> resulted in increased stabilization of HIF-1α and HIF-2α, and RNAi or pharmacologic targeting of p75<sup>NTR</sup> diminished HIF stabilization and HIF-dependent signaling at hypoxia. Consequentially, p75<sup>NTR</sup> inhibition resulted in decreased migration, invasion, and stemness in response to hypoxia, suggesting that p75<sup>NTR</sup> is a central regulator of hypoxia-induced glioma aggressiveness. Together, our findings support the literature that identifies p75<sup>NTR</sup> as a potential therapeutic target in brain tumors.</p>}}, author = {{Tong, Bei and Pantazopoulou, Vasiliki and Johansson, Elinn and Pietras, Alexander}}, issn = {{0014-4827}}, keywords = {{Glioblastoma multiforme; HIF-1α; HIF-2α; Hypoxia; P75 neurotrophin receptor; Stemness}}, language = {{eng}}, month = {{10}}, number = {{1}}, pages = {{122--129}}, publisher = {{Academic Press}}, series = {{Experimental Cell Research}}, title = {{The p75 neurotrophin receptor enhances HIF-dependent signaling in glioma}}, url = {{http://dx.doi.org/10.1016/j.yexcr.2018.08.002}}, doi = {{10.1016/j.yexcr.2018.08.002}}, volume = {{371}}, year = {{2018}}, }