1 – 10 of 1465
- show: 10
- |
- sort: year (new to old)
Close
Embed this list
<iframe src=""
width=""
height=""
allowtransparency="true"
frameborder="0">
</iframe>
- 2023
-
Mark
Combining pharmacophore models derived from DNA-encoded chemical libraries with structure-based exploration to predict Tankyrase 1 inhibitors
Montoya, Alba L ; Glavatskikh, Marta ; Halverson, Brayden J ; Yuen, Lik Hang ; Schüler, Herwig LU
; Kireev, Dmitri
and Franzini, Raphael M
(2023)
In European Journal of Medicinal Chemistry
246.
p.114980-114980
- Contribution to journal › Article
- 2022
-
Mark
Sialic Acid 4-N-Piperazine and Piperidine Derivatives Bind with High Affinity to the P. mirabilis Sialic Acid Sodium Solute Symporter
- Contribution to journal › Article
-
Mark
Large-Scale Crystallographic Fragment Screening Expedites Compound Optimization and Identifies Putative Protein-Protein Interaction Sites
Barthel, Tatjana ; Wollenhaupt, Jan ; Lima, Gustavo M.A. LU
; Wahl, Markus C.
and Weiss, Manfred S.
(2022)
In Journal of Medicinal Chemistry
65(21).
p.14630-14641
- Contribution to journal › Article
-
Mark
The human TRPA1 intrinsic cold and heat sensitivity involves separate channel structures beyond the N-ARD domain
Moparthi, Lavanya LU ; Sinica, Viktor ; Moparthi, Vamsi K LU ; Kreir, Mohamed ; Vignane, Thibaut ; Filipovic, Milos R ; Vlachova, Viktorie and Zygmunt, Peter M LU
(2022)
In Nature Communications
13.
- Contribution to journal › Article
-
Mark
Optimization of N-Piperidinyl-Benzimidazolone Derivatives as Potent and Selective Inhibitors of 8-Oxo-Guanine DNA Glycosylase 1
(2022) In ChemMedChem
- Contribution to journal › Article
-
Mark
Targeting Acute Myelogenous Leukemia Using Potent Human Dihydroorotate Dehydrogenase Inhibitors Based on the 2-Hydroxypyrazolo[1,5- a]pyridine Scaffold : SAR of the Aryloxyaryl Moiety
- Contribution to journal › Article
-
Mark
Discovery of the 4-aminopiperidine-based compound EM127 for the site-specific covalent inhibition of SMYD3
Parenti, Marco Daniele ; Naldi, Marina ; Manoni, Elisabetta ; Fabini, Edoardo ; Cederfelt, Daniela ; Talibov, Vladimir O. LU
; Gressani, Valeria
; Guven, Ummu
; Grossi, Valentina
and Fasano, Candida
, et al.
(2022)
In European Journal of Medicinal Chemistry
243.
- Contribution to journal › Article
-
Mark
Sialic Acid Derivatives Inhibit SiaT Transporters and Delay Bacterial Growth
- Contribution to journal › Article
-
Mark
Design and synthesis of novel 3-triazolyl-1-thiogalactosides as galectin-1, -3 and -8 inhibitors
- Contribution to journal › Article
-
Mark
A hydrophobic patch (PLVIVG; 1481–1486) in the B-domain of factor V-short is crucial for its synergistic TFPIα-cofactor activity with protein S and for the formation of the FXa-inhibitory complex comprising FV-short, TFPIα, and protein S
- Contribution to journal › Article