Drug Target Discovery
1 – 50 of 274
- show: 50
- |
- sort: year (new to old)
Close
Embed this list
<iframe src=" "
width=" "
height=" "
allowtransparency="true"
frameborder="0">
</iframe>
- 2024
-
Mark
G protein-coupled estrogen receptor (GPER)/GPR30 forms a complex with the β1-adrenergic receptor, a membrane-associated guanylate kinase (MAGUK) scaffold protein, and protein kinase A anchoring protein (AKAP) 5 in MCF7 breast cancer cells
(
- Contribution to journal › Article
- 2022
-
Mark
GPR30 in breast cancer - from molecular mechanisms to clinical outcome
2022) In Lund University, Faculty of Medicine Doctoral Dissertation Series(
- Thesis › Doctoral thesis (compilation)
-
Mark
Breast cancer hypoxia in relation to prognosis and benefit from radiotherapy after breast-conserving surgery in a large, randomised trial with long-term follow-up
(
- Contribution to journal › Article
- 2021
-
Mark
Ligand-independent G protein-coupled estrogen receptor/G protein-coupled receptor 30 activity : Lack of receptor-dependent effects of G-1 and 17b-estradiol
(
- Contribution to journal › Article
-
Mark
Mast Cell Proteases Tryptase and Chymase Induce Migratory and Morphological Alterations in Bronchial Epithelial Cells
(
- Contribution to journal › Article
- 2020
-
Mark
Plasma membrane expression of G protein-coupled estrogen receptor (GPER)/G protein-coupled receptor 30 (GPR30) is associated with worse outcome in metachronous contralateral breast cancer
(
- Contribution to journal › Article
- 2019
-
Mark
Human G protein-coupled Receptor 30 (GPR30) is N -glycosylated and N-terminal Domain Asparagine 44 is Required for Receptor Structure and Activity
(
- Contribution to journal › Article
-
Mark
The estrogen receptor coactivator AIB1 is a new putative prognostic biomarker in ER-positive/HER2-negative invasive lobular carcinoma of the breast
(
- Contribution to journal › Article
- 2018
-
Mark
Roles of PDZ-dependent Interactions and N-glycosylation in G Protein-coupled Estrogen Receptor 1 (GPER1)/GPR30-mediated Stimulation of ERK1/2 Activity
(
- Contribution to journal › Published meeting abstract
- 2017
-
Mark
Microvesicle transfer of kinin B1-receptors is a novel inflammatory mechanism in vasculitis
(
- Contribution to journal › Article
-
Mark
G protein-coupled Estrogen Receptor 1 (GPER1)/GPR30 Increases ERK1/2 Activity Through PDZ-dependent and -independent Mechanisms
(
- Contribution to journal › Article
-
Mark
C1-inhibitor decreases the release of vasculitis-like chemotactic endothelial microvesicles
(
- Contribution to journal › Article
-
Mark
AIB1 is a new putative prognostic biomarker in the luminal A and B-like (HER2-negative) classification of invasive lobular carcinoma
(
- Contribution to conference › Abstract
- 2016
-
Mark
Acute hypothalamo-pituitary-adrenal axis response to LPS-induced endotoxemia: expression pattern of kinin type B1 and B2 receptors
(
- Contribution to journal › Article
-
Mark
Bile Acids Protect Expanding Hematopoietic Stem Cells from Unfolded Protein Stress in Fetal Liver.
(
- Contribution to journal › Article
-
Mark
Reduced baseline sensitivity to Maraviroc inhibition among R5 HIV-1 isolates from individuals with severe immunodeficiency.
(
- Contribution to journal › Letter
-
Mark
G protein-coupled Receptor 30 (GPR30) PDZ-dependently and Constitutively Increases ERK1/2 Signaling Through Calcineurin and Kinase Suppressor of Ras 2 (KSR2)
(
- Contribution to journal › Published meeting abstract
- 2015
-
Mark
G Protein-Coupled Estrogen Receptor 1 Mediates Acute Estrogen-Induced Cardioprotection via MEK/ERK/GSK-3β Pathway after Ischemia/Reperfusion.
(
- Contribution to journal › Article
- 2014
-
Mark
The G protein-coupled receptor GPR30 signalosome - A novel G protein-independent mechanism regulating cAMP signaling and receptor trafficking
(
- Thesis › Doctoral thesis (compilation)
-
Mark
G Protein-coupled Receptor 30 (GPR30) Forms a Plasma Membrane Complex With Membrane-associated Guanylate Kinases (MAGUKs) and AKAP5 That Constitutively Inhibits cAMP Production.
(
- Contribution to journal › Article
-
Mark
Lack of G protein-coupled estrogen receptor (GPER) in the plasma membrane is associated with excellent long-term prognosis in breast cancer.
(
- Contribution to journal › Article
- 2013
-
Mark
G-protein-coupled receptor 30 interacts with receptor activity-modifying protein 3 and confers sex-dependent cardioprotection
(
- Contribution to journal › Article
-
Mark
Kinin B1 receptor homo-oligomerization is required for receptor trafficking to the cell surface.
(
- Contribution to journal › Article
-
Mark
G protein-coupled estrogen receptor is apoptotic and correlates with increased distant disease-free survival of estrogen receptor-positive breast cancer patients.
(
- Contribution to journal › Article
-
Mark
Contact allergy from disperse dyes in textiles-a review.
(
- Contribution to journal › Article
- 2012
-
Mark
The G protein-coupled oestrogen receptor 1 agonist G-1 disrupts endothelial cell microtubule structure in a receptor-independent manner.
(
- Contribution to journal › Article
-
Mark
Dual R3R5 tropism characterizes cerebrospinal fluid HIV-1 isolates from individuals with high cerebrospinal fluid viral load
(
- Contribution to journal › Article
-
Mark
17 beta-Estradiol induces nongenomic effects in renal intercalated cells through G protein-coupled estrogen receptor 1
(
- Contribution to journal › Article
- 2011
-
Mark
G protein-coupled oestrogen receptor 1 (GPER1)/GPR30: a new player in cardiovascular and metabolic oestrogenic signalling
(
- Contribution to journal › Scientific review
-
Mark
Serum gastrin and gastric enterochromaffin-like cells during estrous cycle, pregnancy and lactation, and in response to estrogen-like agents in rats
(
- Contribution to journal › Article
-
Mark
Textile Dyes Disperse Orange 1 and Yellow 3 Contain More Than One Allergen As Shown by Patch Testing with Thin-Layer Chromatograms
(
- Contribution to journal › Article
-
Mark
G Protein-Coupled Estrogen Receptor 1 (GPER1)/GPR30 Localizes in the Plasma Membrane and Trafficks Intracellularly on Cytokeratin Intermediate Filaments.
(
- Contribution to journal › Article
-
Mark
Insulinotropic and Antidiabetic Effects of 17{beta}-Estradiol and the GPR30 Agonist G-1 on Human Pancreatic Islets.
(
- Contribution to journal › Article
-
Mark
Abnormally decreased NO and augmented CO production in islets of the leptin-deficient ob/ob mouse might contribute to explain hyperinsulinemia and islet survival in leptin-resistant type 2 obese diabetes.
(
- Contribution to journal › Article
-
Mark
The GPER1 Agonist G-1 Attenuates Endothelial Cell Proliferation by Inhibiting DNA Synthesis and Accumulating Cells in the S and G2 Phases of the Cell Cycle.
(
- Contribution to journal › Article
-
Mark
New topics in bradykinin research.
(
- Contribution to journal › Article
-
Mark
P4-09-02: G Protein-Coupled Estrogen Receptor 1 Positively Correlates with Estrogen Receptor a Expression and Increased Distant Disease-Free Survival of Breast Cancer Patients.
(
- Contribution to journal › Published meeting abstract
- 2010
-
Mark
Defective secretion of islet hormones in chromogranin-B deficient mice.
(
- Contribution to journal › Article
-
Mark
Proghrelin peptides: Desacyl ghrelin is a powerful inhibitor of acylated ghrelin, likely to impair physiological effects of acyl ghrelin but not of obestatin A study of pancreatic polypeptide secretion from mouse islets.
(
- Contribution to journal › Article
-
Mark
Gastrin release: Antrum microdialysis reveals a complex neural control.
(
- Contribution to journal › Article
-
Mark
Gastrin response to candidate messengers in intact conscious rats monitored by antrum microdialysis.
(
- Contribution to journal › Article
-
Mark
ADP mediates inhibition of insulin secretion by activation of P2Y13 receptors in mice.
(
- Contribution to journal › Article
- 2009
-
Mark
Low gastric acid and high plasma gastrin in high-anxiety Wistar Kyoto rats
(
- Contribution to journal › Article
-
Mark
Activation Of The Putative Estrogen Receptor Gpr30 Attenuates Endothelial Cell Dna Synthesis
2009) 14th Annual Meeting of the European-Council-for-Cardiovascular-Research In Hypertension 54(5). p.1186-1186(
- Contribution to journal › Published meeting abstract
-
Mark
Neutrophil-derived proteinase 3 induces kallikrein-independent release of a novel vasoactive kinin
(
- Contribution to journal › Published meeting abstract
-
Mark
Activation of TAFI on the Surface of Streptococcus pyogenes Evokes Inflammatory Reactions by Modulating the Kallikrein/Kinin System
(
- Contribution to journal › Article
-
Mark
Palmitate-stimulated hormone secretion in relation to GPR40 expression in pancreatic islets of spontaneous obesity and type 2 diabetes in rats
2009) 45th Annual Meeting of the European-Association-for-the-Study-of-Diabetes In Diabetologia 52(Suppl. 1). p.405-405(
- Contribution to journal › Published meeting abstract
-
Mark
Islet-cell secretion of pancreatic polypeptide in response to ghrelin and obestatin acting on distinct receptors
2009) 45th Annual Meeting of the European-Association-for-the-Study-of-Diabetes In Diabetologia 52(Suppl 1). p.605-605(
- Contribution to journal › Published meeting abstract
-
Mark
G protein-coupled receptor regulation: The role of protein interactions and receptor trafficking
(
- Thesis › Doctoral thesis (compilation)
-
Mark
The role of the G protein-coupled receptor GPR30 in the effects of estrogen in ovariectomized mice
(
- Contribution to journal › Article