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- 2024
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Mark
Discovery of the Selective and Orally Available Galectin-1 Inhibitor GB1908 as a Potential Treatment for Lung Cancer
2024) In Journal of Medicinal Chemistry(
- Contribution to journal › Article
- 2023
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Mark
Fluorescently Guided Optical Photothermal Infrared Microspectroscopy for Protein-Specific Bioimaging at Subcellular Level
(
- Contribution to journal › Article
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Mark
Ligand Sulfur Oxidation State Progressively Alters Galectin-3-Ligand Complex Conformations To Induce Affinity-Influencing Hydrogen Bonds
(
- Contribution to journal › Article
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Mark
Strong Binding of C-Glycosylic1,2-Thiodisaccharides to Galectin-3─Enthalpy-Driven Affinity Enhancement by Water-Mediated Hydrogen Bonds
(
- Contribution to journal › Article
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Mark
Discovery of Selective and Orally Available Galectin-1 Inhibitors
(
- Contribution to journal › Article
- 2018
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Mark
Elucidation of Hydrogen Bonding Patterns in Ligand-Free, Lactose- and Glycerol-Bound Galectin-3C by Neutron Crystallography to Guide Drug Design
(
- Contribution to journal › Article
- 2017
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Mark
Fragment-Based Discovery and Optimization of Enzyme Inhibitors by Docking of Commercial Chemical Space
(
- Contribution to journal › Article
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Mark
Class II Phosphoinositide 3-Kinases as Novel Drug Targets
(
- Contribution to journal › Scientific review
- 2016
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Mark
Chiral Dihydrobenzofuran Acids Show Potent Retinoid X Receptor-Nuclear Receptor Related 1 Protein Dimer Activation.
(
- Contribution to journal › Article
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Mark
Experimental Active-Site Mapping by Fragments - Hot Spots Remote from the Catalytic Center of Endothiapepsin
2016) In Journal of Medicinal Chemistry(
- Contribution to journal › Article
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Mark
Studies on Aryl-Substituted Phenylalanines: Synthesis, Activity, and Different Binding Modes at AMPA Receptors
(
- Contribution to journal › Article
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Mark
Inhibitors of the Cysteine Synthase CysM with Antibacterial Potency against Dormant Mycobacterium tuberculosis
(
- Contribution to journal › Article
- 2015
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Mark
Synthesis and Biological Evaluation of Second-Generation Tropanol-Based Androgen Receptor Modulators
(
- Contribution to journal › Article
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Mark
Disubstituted Bis-THF Moieties as New P2 Ligands in Nonpeptidal HIV-1 Protease Inhibitors (II)
(
- Contribution to journal › Article
- 2014
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Mark
Synthesis of P1 '-Functionalized Macrocyclic Transition-State Mimicking HIV-1 Protease Inhibitors Encompassing a Tertiary Alcohol
(
- Contribution to journal › Article
- 2013
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Mark
Tuning the Preference of Thiodigalactoside- and Lactosamine-Based Ligands to Galectin-3 over Galectin-1
(
- Contribution to journal › Article
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Mark
Design and Synthesis of P1-P3 Macrocyclic Tertiary-Alcohol-Comprising HIV-1 Protease Inhibitors
(
- Contribution to journal › Article
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Mark
Synthesis, pharmacological and structural characterization, and thermodynamic aspects of GluA2-positive allosteric modulators with a 3, 4-dihydro-2 H-1, 2, 4-benzothiadiazine 1, 1-dioxide scaffold
(
- Contribution to journal › Article
-
Mark
HAHAHA, HEHEHE, HIHIHI, or HKHKHK : influence of position and composition of histidine containing tags on biodistribution of [(99m)Tc(CO)3](+)-labeled affibody molecules
(
- Contribution to journal › Article
- 2012
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Mark
Synthesis, X-ray Analysis, and Biological Evaluation of a New Class of Stereopure Lactam-Based HIV-1 Protease Inhibitors
(
- Contribution to journal › Article
- 2011
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Mark
Difluoromethylbenzoxazole Pyrimidine Thioether Derivatives: A Novel Class of Potent Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors
(
- Contribution to journal › Article
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Mark
Molecular Wipes: Application to Epidemic Keratoconjuctivitis
(
- Contribution to journal › Article
- 2008
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Mark
Galectin-inhibitory thiodigalactoside ester derivatives have antimigratory effects in cultured lung and prostate cancer cells.
(
- Contribution to journal › Article
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Mark
Arginine Binding Motifs: Design and Synthesis of Galactose-Derived Arginine Tweezers as Galectin-3 Inhibitors.
(
- Contribution to journal › Article
- 2007
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Mark
Synthesis and transfection efficiencies of new lipophilic polyamines
(
- Contribution to journal › Article
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Mark
Probing Molecular Interactions within Class II MHC A(q)/Glycopeptide/T-Cell Receptor Complexes Associated with Collagen-Induced Arthritis.
(
- Contribution to journal › Article
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Mark
Quantitative Structure-Activity Relationship of Peptides Binding to the Class II Major Histocompatibility Complex Molecule A(q) Associated with Autoimmune Arthritis.
(
- Contribution to journal › Article
- 2006
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Mark
Selective antiproliferative activity of hydroxynaphthyl-beta-D-xylosides
(
- Contribution to journal › Article
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Mark
Ligand affinities predicted with the MM/PBSA method: Dependence on the simulation method and the force field
(
- Contribution to journal › Article
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Mark
4-quinolone derivatives: High-affinity ligands at the benzodiazepine site of brain GABA(A) receptors. synthesis, pharmacology, and pharmacophore modeling
(
- Contribution to journal › Article
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Mark
Prediction of activation energies for hydrogen abstraction by cytochrome P450
(
- Contribution to journal › Article
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Mark
Novel selective orally active CRTH2 antagonists for allergic inflammation developed from in silico derived hits
(
- Contribution to journal › Article
- 2005
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Mark
Light-Induced Anticancer Activity of [RuCl2(DMSO)4] Complexes
(
- Contribution to journal › Article
- 2002
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Mark
Refinement and evaluation of a pharmacophore model for flavone derivatives binding to the benzodiazepine site of the GABA(A) receptor
(
- Contribution to journal › Article
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Mark
Methanocarba modification of uracil and adenine nucleotides: High potency of northern ring conformation at P2Y(1), P2Y(2), P2Y(4), and P2Y(11) but not P2Y(6) receptors
(
- Contribution to journal › Article
-
Mark
Azapeptides structurally based upon inhibitory sites of cystatins as potent and selective inhibitors of cysteine proteases
(
- Contribution to journal › Article
- 2000
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Mark
Computational predictions of binding affinities to dihydrofolate reductase: synthesis and biological evaluation of methotrexate analogues
(
- Contribution to journal › Article